安池 修之 教授

研究業績一覧
  1. Synthesis and optical properties of N-arylnaphtho- and anthra[2,3-d]oxazol-2-amines. Y. Murata, M. Kawakubo, A. Maruyama, M. Matsumura and S. Yasuike, Molecules, 30, 319 (2025).
  2. Synthesis of sulfenamides from benzoazole-2-thiones with primary and secondary amines using triphenylbismuth dichloride-mediated S-N bond formation reaction. A. Koyanagi, Y. Murata, M. Matsumura and S. Yasuike, Asian J. Org. Chem., 13, e202400138 (2024).
  3. Bismuth(III)-catalyzed regioselective selenation of Indoles with diaryl diselenides: synthesis of 3-selanylindoles. M. Matsumura, A. Umeda, Y. Sumi, N. Aiba, Y. Murata and S. Yasuike, Molecules, 29, 3227 (2024).
  4. Synthesis of tetracyclic benzazole-condensed quinazolinones through triphenylbismuth dichloride assisted cyclodesulfurization. A. Koyanagi, Y. Murata, C. Takeshita, Y. Kato, M. Matsumura and S. Yasuike. Synthesis, 56, 2109-2117 (2024).
  5. Novel mono substituted pyridoimidazoisoquinoliniums via a silver-catalyzed intramolecular cyclization and their applications in cellular imaging. M. Kawakubo, Y. Inoh, Y. Murata, M. Matsumura, T. Furuno, and S. Yasuike. RSC Adv., 14, 9758-9762 (2024).
  6. Synthesis and intracellular localization of 5,6-disubsutituted pyrido[1′,2′;2,3]imidazo[5,1-a]isoquinolinium iodides. M. Kawakubo, Y. Inoh, Y. Inaguma, R. Kokubugata, Y. Murata, M. Matsumura, T. Furuno and S. Yasuike. ChemistrySelect, 8, e202303017 (2023).
  7. Palladium-Catalyzed Cross-coupling Reaction of Bis(cyclopentadienyl)diaryltitaniums with Terminal Alkynes. Y. Murata, Y. Nishi, M. Matsumura and S. Yasuike. Reactions, 4, 657-666 (2023).
  8. Copper-catalyzed three-component reaction of pyrazol-3-ones (antipyrine), triarylbismuthines, and selenium: Synthesis of 4-selanylpyrazol-3-ones. M. Matsumura, A. Nakamura, A. Yanagida, Y. Murata and S. Yasuike. Tetrahedron, 142, 133526 (2023).
  9. Palladium-catalyzed C-H arylation of quinoxalin-2(1H)-ones with triarylantimony difluorides. M. Matsumura, H. Nojima, Y. Kitamura, Y. Murata, and S. Yasuike, J. Organometalic. Chem., 989, 122639 (2023).
  10. Sb-Phenyl-N-methyl-5,6,7,12-tetrahydrodibenz[c,f][1,5]azastibocine induces perlecan core protein synthesis in cultured vascular endothelial cells. T. Hara, T. Konishi, S. Yasuike, Y. Fujiwara, C. Yamamoto and T. Kaji, Int. J. Mol. Sci., 24, 3656-546 (2023).
  11. Triphenylbismuth dichloride inhibits human glyoxalase I and induces cytotoxicity in cultured cancer cell lines. R. Takasawa, A. Jona, M. Inoue, M. Azuma, H. Akahane, Y. Ueno, Y. Nakagawa, R. Chimori, Y. Mano, Y. Murata, S. Yasuike and T. Kaji, J. Toxicol. Sci., 47, 539-546 (2022).
  12. One-pot synthesis of 2-arylated and 2-alkylated benzoxazoles and benzimidazoles based on triphenylbismuth dichloride-promoted desulfurization of thioamides. A. Koyanagi, Y. Murata, S. Hayakawa, M. Matsumura and S. Yasuike, Beilstein J. Org. Chem., 18, 1479-1487 (2022).
  13. Synthesis of novel 5-iodopyrido[1',2';2,3]imidazo[5,1-a]isoquinolinium iodides from 2-(2-ethynylphenyl)imidazo[1,2-a]pyridines via iodocyclization. M. Kawakubo, Y. Inaguma, Y. Murata, M. Matsumura and S. Yasuike, Tetrahedron Lett., 105, 154054 (2022).
  14. Synthesis of novel alkynyl imidazopyridinyl selenides: copper-catalyzed tandem selenation of selenium with 2-arylimidazo[1,2-a]pyridines and terminal alkynes. M. Matsumura, K. Tsukada, K. Sugimoto, Y. Murata and S. Yasuike, Beilstein J. Org. Chem., 18, 863-871 (2022).
  15. Silver-catalyzed three-component reaction of uracils, arylboronic acids, and selenium: synthesis of 5-arylselanyluracils. Y. Murata, S. Tsuchida, R. Nezaki, Y. Kitamura, M. Matsumura and S. Yasuike, RSC Adv., 12, 14502, (2022).
  16. Synthesis and optical properties of azuleno[1,2-b]benzothiophene and selenophene. M. Matsumura, T. Kamiya, M. Kawakubo, Y. Hayashi, T. Hyodo, Y. Murata, K. Yamaguchi and S. Yasuike, Heterocycles, 105, 337-342, (2022).
  17. Effects of substitution on cytotoxicity of diphenyl ditelluride in cultured vascular endothelial cells. T. Hara, T. Okazaki, T. Hashiya, K. Nozawa, S. Yasuike, J. Kurita, C. Yamamoto, N. Hamada and T. Kaji, Int. J. Mol. Sci., 22, 10520 (2021).
  18. Copper-catalyzed C−H selenation of 2-substituted benzo[b]furans with diaryl diselenides: Synthesis of 2-substituted 3-selanylbenzo[b]furan derivatives. Y. Murata, N. Otake, M. Sano, M. Matsumura and S. Yasuike, Asian J. Org. Chem., 10, 2975-2981 (2021).
  19. Construction of dibenzo[d,f][1,3]oxazepine skeleton from 2'-amino-2-hydroxybiphenyl and via iodine-mediated cyclodesulfurization.isothiocyanates. Y. Murata, M. Izawa, A. Koyanagi, Y. Hayashi, T. Hyodo, M. Matsumura, K. Yamaguchi and S. Yasuike, Tetrahedron Lett., 73, 153142 (2021).
  20. Synthesis, structural characterization, and optical properties of benzo[f]naphtho[2,3-b]phosphoindoles. M. Matsumura, T. Teramoto, M. Kawakubo, M. Kawahata, Y. Murata, K. Yamaguchi, M. Uchiyama and S. Yasuike, Beilstein J. Org. Chem., 17, 671-677 (2021).
  21. Synthesis, structural characterization, and optical properties of benzene-fused tetracyclic and pentacyclic stiboles. M. Matsumura, Y. Matsuhashi, M. Kawakubo, T. Hyodo. Y. Murata, M. Kawahata, K. Yamaguchi and S. Yasuike, Molecules, 26, 222 (2021).
  22. Palladium-catalyzed C―H arylation of benzofurans with triarylantimony difluorides for the synthesis of 2-arylbenzofurans. Y. Kitamura, Y. Murata, M. Iwai, M. Matsumura and S. Yasuike, Molecules, 26, 97 (2021).
  23. Pd-catalyzed oxidative Heck-type arylation of vinyl ketones, alkenes, and acrylates with Sb-aryltetrahydrodibenz[c,f][1,5]azastibocines. Y. Murata, N. Kakusawa, Y. Arakawa, Y. Hayashi, S. Morinaga, M. Ueda, T. Hyodo, M. Matsumura, K. Yamaguchi, J. Kurita and S. Yasuike, J. Organomet. Chem., 928, 121545 (2020).
  24. Liebeskind-Srogl-type cross-coupling reaction of azole-2-thiones with triarylbismuthines: Synthesis of 2-arylazoles. Y. Murata, A.Terazoe, M. Kiba, Y. Kitamura, M. Matsumura and S. Yasuike, Tetrahedron Lett., 61, 152152 (2020).
  25. Synthesis of nitriles via the iodine-mediated dehydrosulfurization of thioamides. Y. Murata, H. Iwasa, M. Matsumura and S. Yasuike, Chem. Pharm. Bull., 68, 679-681 (2020).
  26. Synthesis and anticancer activity of bis(2-arylimidazo[1,2-a]pyridin-3-yl) selenides and diselenides: the copper-catalyzed tandem C―H selenation of 2-arylimidazo[1,2-a]pyridine with selenium. M. Matsumura, T. Takahashi, H. Yamauchi, S. Sakuma, Y. Hayashi, T. Hyodo, T. Obata, K. Yamaguchi, Y. Fujiwara and S. Yasuike, Beilstein J. Org. Chem., 16, 1075-1083 (2020).
  27. Cascade synthesis of 4-arylcoumarins: Pd-catalyzed arylations and cyclizations with (E)-ethyl 3-(2-hydroxyaryl)acrylates and triarylantimony difluorides. Y. Kitamura, M. Matsumura, Y. Kato, Y. Murata and S. Yasuike, Eur. J. Org. Chem., 2020, 1652-1657 (2020).
    Selected as Very Important Paper (VIP)
  28. Synthesis of 2-(arylsulfenyl)azoles by copper-catalyzed S-arylation of azole-2-thiones with triarylbismuthines. Y. Murata, S. Asano, R. Kato, Y. Kitamura, M. Matsumura and S. Yasuike, Catal. Commun., 132, 105808 (2019).
  29. Intracellular accumulation-independent cytotoxicity of pentavalent organoantimony compounds in cultured vascular endothelial cells. T. Hara, S. Nakano, Y. Kitamura, C. Yamamoto, S. Yasuike and T. Kaji, J. Toxicol. Sci., 44, 845-848 (2019).
  30. 13-(2-Methylbenzyl)berberine is a more potent inhibitor of MexXY-dependent aminoglycoside resistance than berberine. K. Kotani, M. Matsumura, Y. Morita, J. Tomida, R. Kutsuna, K. Nishino, S. Yasuike and Y. Kawamura, Antibiotics, 8, 212-224 (2019).
  31. Synthesis of benzo[d]imidazo[2,1-b]benzoselenoazoles: Cs2CO3-mediated cyclization of 1-(2-bromoaryl)benzimidazoles with selenium. M. Matsumura, Y. Kitamura, A. Yamauchi, Y. Kanazawa, Y. Murata, T. Hyodo, K. Yamaguchi and S. Yasuike, Beilstein J. Org. Chem., 15, 2029-2035 (2019).
  32. Efficient synthesis, structural characterization, and optical properties of 6H-dibenzo[b,h]carbazole and its derivatives. M. Matsumura, M. Kawahata, A. Muranaka, M. Hiraiwa, K. Yamaguchi, M. Uchiyama and S. Yasuike, Eur. J. Org. Chem., 2019, 3788-3793 (2019).
  33. Possible mechanisms underlying transcriptional induction of metallothionein informs by tris(pentafluorophenyl)stibane, tris(pentafluorophenyl)arsane, and tris(pentafluorophenyl)phosohane in cultured bovine aortic endothelial cells. T. Fujie, F. Takenaka, E. Yoshida, S. Yasuike, Y. Fujiwara, Y. Shinkai, Y. Kumagai, C. Yamamoto and T. Kaji, J. Toxicol. Sci., 44, 327-333 (2019).
  34. Copper-catalyzed three-component reaction of ethynylstibanes, organic azides, and selenium: A simple and efficient synthesis of novel selenides and diselenides having 1,2,3-triazole rings. M. Yamada, M. Matsumura, E. Sakaki, S.-y. Yen, M. Kawahata, T. Hyodo, K. Yamaguchi, Y. Murata and S. Yasuike, Tetrahedron, 75, 1406-1414 (2019).
  35. Visible-light-promoted Se-arylation of diaryl diselenides with 2-phenylimidazopyridines in the presence of ammonium iodide: Synthesis of 2-phenyl-3-(arylselanyl)imidazo[1,2-a]pyridines. Y. Murata, K. Kanasaki, K. Kondo, N. Kakusawa, M. Matsumura and S. Yasuike, Heterocycles, 99, 596-603 (2019).
  36. Pd-catalyzed β-selective C-H arylation of thiophenes with triarylantimony difluorides. Y. Kitamura, Y. Murata, A. Oguri, M. Matsumura, N. Kakusawa, H. Naka and S. Yasuike, Asian J. Org. Chem., 8, 138-143 (2019).
  37. Structure-activity relationship of [1,5]azastibocines in cytotoxicity to vascular endothelial cells. T. Hara, Y. Nonaka, S. Yasuike, T. Kaji and C. Yamamoto, J. Toxicol. Sci., 43, 735-740 (2018).
  38. Copper-catalyzed cross-coupling reactions of 5-stibano-1,2,3-triazoles with bromoalkynes under aerobic conditions: Synthesis of 5-alkynyl-1,2,3-triazoles. M. Yamada, D. Matsuura, M. Hasegawa, Y. Murata, N. Kakusawa, M. Matsumura and S. Yasuike, J. Organomet. Chem., 871, 79-85 (2018).
  39. Synthesis of 2-aryl-3-(arylselanyl)imidazo[1,2-a]pyridines: copper-catalyzed one-pot two-step Se-Arylation of selenium with imdazopyridines and triarylbismuthanes. K. Kondo, M. Matsumura, K. Kanasaki, Y. Murata, N. Kakusawa and S. Yasuike, Synthesis, 50, 2200-2210 (2018).
    Highlighted as a Front Cover
  40. One-pot reaction for the synthesis of N-substituted 2-aminobenzoxazoles using triphenylbismuth dichloride as cyclodesulfurization reagent. Y. Murata, N. Matsumoto, M. Miyata, Y. Kitamura, N. Kakusawa, M. Matsumura and S. Yasuike, J. Organomet. Chem., 859, 18-23 (2018).
  41. Synthesis, antitumor activity, and cytotoxicity of 4-substituted 1-benzyl-5-diphenylstibano-1H-1,2,3-triazoles. M. Yamada, T. Takahashi, M. Hasegawa, M. Matsumura, K. Ono, R. Fujimoto, Y. Kitamura, Y. Murata, N. Kakusawa, M. Tanaka, T. Obata, Y. Fujiwara and S. Yasuike, Bioorg. Med. Chem. Lett., 28, 152-154 (2018).
  42. Synthesis of fully functionalized 5-selanyl-1,2,3-triazoles: Copper-catalyzed three-component reaction of ethynylstibanes, organic azides, and diaryl diselenides. M. Yamada, M. Matsumura, F. Takino, Y. Murata, Y. Kurata, M. Kawahata, K. Yamaguchi, N. Kakusawa and S. Yasuike, Eur. J. Org. Chem., 2018, 170-177 (2018).
  43. Microwave-assisted debromination of α-bromoketones with triarylstibanes in water. Y. Murata, Y. Sugawara, M. Matsumura, N. Kakusawa and S. Yasuike, Chem. Pharm. Bull., 65, 1081-1084 (2017).
  44. Synthesis and photophysical properties of novel benzophospholo[3,2-b]indole derivatives. M. Matsumura, M. Yamada, A. Muranaka, M. Kanai, N. Kakusawa, D. Hashizume, M. Uchiyama and S. Yasuike, Beilstein J. Org. Chem., 13, 2304-2309 (2017).
  45. Synthesis of 5-organostibano-1H-1,2,3-triazoles by Cu-catalyzed azide-alkyne cycloaddition and their application in the acyl-induced deantimonation for the preparation of fully substituted 5-acyl-1,2,3-triazoles. M. Yamada, Y. Murata, M. Matsumura, M. Kawahata, K. Saito, N. Kakusawa, K. Yamaguchi and S. Yasuike, J. Fluor. Chem., 199, 1-6 (2017).
  46. A versatile synthesis of triarylantimony difluorides by fluorination of triarylstibanes with nitrosyl tetrafluoroborate and their antitumor activity. Y. Kitamura, M. Matsumura,Y. Murata, M. Yamada, N. Kakusawa, M. Tanaka, H. Okabe, H. Naka, T. Obata and S. Yasuike, Tetrahedron, 73, 2614-2622 (2017).
  47. Anti-inflammatory effect of JBP485 on Dextran Sulfate Sodium-induced Colitis in Mice. S. Horibe, S. Kawauchi, S. Yasuike, S. Mizuno, I. Kato and Y. Rikitake, J. Biomed., 2, 101-108 (2017).
  48. Antimony-lithium exchange reaction: Synthesis of 1,4,5-trisubstituted-1,2,3-triazoles by triazolyllithium with electrophiles. M. Yamada, M. Matsumura, M. Kawahata, Y. Murata, N. Kakusawa, K. Yamaguchi and S. Yasuike, J. Organomet. Chem., 834, 83-87 (2017).
  49. Copper-catalyzed tandem cyclization of 2-(2-iodophenyl)imidazo[1,2-a]pyridine derivatives with selenium: Synthesis of benzo[b]selenophene-fused imidazo[1,2-a]pyridines. M. Matsumura, Y. Sakata, A. Iwase, Y. Kawahata, M. Kitamura, Y. Murata, N. Kakusawa, K. Yamaguchi and S. Yasuike, Tetrahedron Lett., 57, 5484-5488 (2016).
  50. General synthesis, structure, and optical properties of benzothiophene-fused benzoheteroles containing Group 15 and 16 elements. M. Matsumura, A. Muranaka, R. Kurihara, M. Kanai, K. Yoshida, N. Kakusawa, D. Hashizume, M. Uchiyama and S. Yasuike, Tetrahedron, 72, 8085-8090 (2016).
  51. Transcriptional induction of metallothionein by tris(pentafluorophenyl)stibane in cultured bovine aortic endothelial cells. T. Fujie, M. Murakami, E. Yoshida, S. Yasuike, T. Kimura, Y. Fujiwara, C. Yamamoto and T. Kaji, Int. J. Mol. Sci., 17, 1381 (2016).
  52. Copper-catalyzed [3+2] cycloaddition of (phenylethynyl)di-p-tolylstibane with organic azides. M. Yamada, M. Matsumura, Y. Uchida, M. Kawahata, Y. Murata, N. Kakusawa, K. Yamaguchi and S. Yasuike, Beilstein J. Org. Chem., 12, 1309-1313. (2016).
  53. Synthesis of unsymmetrical diaryl selenides: copper-catalyzed Se-arylation of diaryl diselenides with triarylbismuthanes. M. Matsumura, K. Shibata, S. Ozeki, M. Yamada, Y. Murata, N. Kakusawa and S. Yasuike, Synthesis, 48, 730-736 (2016).
  54. Synthesis, structural characterization and antitumor activity of 2-(di-p-tolylstibano)- and 2-(di-p-tolylbismuthano)-N-p-tolylbenzamide. T. Obata, M. Matsumura, M. Kawahata, S. Hoshino, M. Yamada, Y. Murata, N. Kakusawa, K. Yamaguchi, M. Tanaka and S. Yasuike, J. Organomet. Chem., 807, 17-21 (2016).
  55. Synthesis of 2-arylquinoxalines: triarylstibane catalyzed oxidative cyclization of α-hydroxy ketones with 1,2-diamines under aerobic conditions. M. Matsumura, R. Takada, Y. Ukai, M. Yamada, Y. Murata, N. Kakusawa and S. Yasuike, Heterocycles, 93, 75-83 (2016).
    Highlighted in SYNFACTS, 2016, 12 (2), 0128.
  56. Simple and efficient copper-catalyzed synthesis of symmetrical diaryl selenides from triarylbismuthanes and selenium under aerobic conditions. M. Matsumura, H. Kumagai, Y. Murata, N. Kakusawa and S. Yasuike, J. Organomet. Chem., 807, 11-16 (2016).
  57. Palladium-catalyzed cross-coupling reactions of triarylbismuthanes with terminal alkynes under aerobic conditions. M. Matsumura, M. Yamada, T. Tsuji, Y. Murata, N. Kakusawa and S. Yasuike, J. Organomet. Chem., 794, 70-75 (2015).
  58. Preparation of acylthiophenes by iron(III) chloride catalyzed reactions of tris(2-thienyl)stibanes with acyl chlorides. N. Kakusawa, Y. Nakagawa, Y. Toshima, S. Yasuike and J. Kurita, Heterocycles, 91, 1170-1175 (2015).
  59. Synthesis of arylboronates by boron-induced ipso-deantimonation of triarylstibanes with boron trihalides and its application in one-pot two-step transmetallation/cross-coupling reactions. S. Yasuike, K. Nakata, W. Qin, M. Matsumura, N. Kakusawa and J. Kurita, J. Organomet. Chem., 788, 9-16 (2015).
  60. The cytotoxicity of organobismuth compounds with certain molecular structures can be diminished by replacing the bismuth atom with an antimony atom in the molecules. K. Kohri, E. Yoshida, T. Fujie, S. Yasuike, C. Yamamoto and T. Kaji, J. Toxicol. Sci., 40, 321-327 (2015).
    Pfizer Highly Cited Paper Award in The Japanese Society of Toxicology.
  61. Comparative cytotoxicity of triphenylstibane and fluorine-substituted triarylpnictogens in cultured vascular endothelial cells. M. Murakami, T. Fujie, M. Matsumura, E. Yoshida, C. Yamamoto, Y. Fujiwara, S. Yasuike and T. Kaji, Fundam. Toxicol. Sci., 2, 61-66 (2015).
  62. Pd-Catalyzed P-arylation of triarylantimony dicarboxylates with dialkyl H-phosphites without a base: Synthesis of arylphosphonates. M. Matsumura, Y. Dong, N. Kakusawa and S. Yasuike, Chem. Pharm. Bull., 63, 130-133 (2015).
  63. Synthesis and structural characterization of a novel organotellurium compound: Dinaphtho[2,3-b;2’,3’-d]tellurophene. M. Matsumura, A. Muranaka, N. Kakusawa, J. Kurita, D. Hashizume, M. Uchiyama and S. Yasuike, Heterocycles, 90, 121-125 (2015).
  64. Simple base-free Miyaura-type borylation of triarylantimony diacetates with tetra(alkoxo)diborons under aerobic conditions. S. Yasuike, Y. Dong, N. Kakusawa, M. Matsumura and J. Kurita, J. Organomet. Chem., 765, 80-85 (2014).
  65. Syntheses of novel dibenzo[d,f]heteronins incorporating group 15 and 16 heavier elements. S. Yasuike, S. Tsukada, N. Kakusawa, T. Tsuchiya and J. Kurita, Heterocycles, 86, 941-945 (2012).
  66. A novel organobismuth compound, 1-[(2-di-p-tolylbismuthanophenyl)diazenyl]pyrrolidine, induces apoptosis in the human acute promyelocytic leukemia cell line NB4 via reactive oxygen species. K. Onishi, M. Douke, T. Nakamura, Y. Ochiai, N. Kakusawa, S. Yasuike, J. Kurita, C. Yamamoto, M. Kawahata, K. Yamaguchi and T. Yagura, J. Inorg. Biochem., 117, 77-84 (2012).
  67. Bis(L-cysteinato)zincate(II) as a coordination compound that specifically induces metallothionein gene transcription without inducing cell-stress-related gene transcription. T. Kimura, K. Yoshida, C. Yamamoto, M. Suzuki, T. Uno, M. Isobe, H. Naka, S. Yasuike, M. Satoh, T. Kaji and M. Uchiyama, J. Inorg. Biochem., 117, 140-148 (2012).
  68. Aluminepin: Aluminum analogues of borepin and gallepin. K, Yoshida, T. Furuyama, C. Wang, A. Muranaka, D. Hashizume, S. Yasuike and M. Uchiyama, J. Org. Chem., 77, 729-732 (2012).
  69. Simple and efficient copper-catalyzed S-arylation of diaryl disulfides with triarylbismuthanes under aerobic conditions. S. Yasuike, M. Nishioka, N. Kakusawa and J. Kurita, Tetrahedron Lett., 52, 6403-6406 (2011).
  70. [2-(N,N-Dimethylaminomethyl)phenyl]bis(4-methylphenyl)bismuthane. M. Kawahata, S. Yasuike, I. Kinebuchi, K. Yamaguchi and J. Kurita, Acta Cryst. E, E67, m25 (2011).
  71. Rhodium-catalyzed 1,2-addition of Sb-phenyl-1,5-azastibocines to functionalized aldehydes. N. Kakusawa, S. Yasuike and J. Kurita, Heterocycles, 80, 163-168 (2010).
  72. Reaction mechanism for the LiCl-mediated directed zinc insertion: A computational and experimental study. C. Liu, X. Wang, T. Furuyama, S. Yasuike, A. Muranaka, K. Morokuma and M. Uchiyama, Chem. Eur. J., 16, 1780-1784 (2010).
  73. Synthesis of optically active P-chirogenic ferrocene-fused benzophosphole by diastereoselective intramolecular cyclization of phosphanylferrocene derivatives. S. Yasuike, J. Hagiwara, H. Danjo, M. Kawahata, N. Kakusawa, K. Yamaguchi and Jyoji Kurita, Heterocycles, 78, 3001-3010 (2009).
  74. Copper- and base-free Sonogashira-type cross-coupling reaction of triarylantimony dicarboxylates with terminal alkynes under an aerobic condition. X. Wang, W. Qin, N. Kakusawa, S. Yasuike and J. Kurita, Tetrahedron Lett., 50, 6293-6297 (2009).
  75. Pentavalent organoantimony compounds as mild N-arylating agents for amines: Cu-mediated Ullmann-type N-arylation with tetraarylantimony(V)acetates. W. Qin, N. Kakusawa, Y. Wu, S. Yasuike and J. Kurita, Chem. Pharm. Bull., 57, 436-438 (2009).
  76. Gilman-type versus Lipshutz-type reagents: competition in lithiocuprate chemistry. J. Haywood, J. V. Morey, A. E. H. Wheatly, C-Y. Liu, S. Yasuike, J. Kurita, M. Uchiyama, P. Raithby, Organometallics, 28, 38-41 (2009).
  77. Synthesis and thermal stability of 3-substituented-3-benzostibepines. S. Yasuike, M. Ikoma, N. Kakusawa, T. Tsuchiya and J. Kurita, Heterocycles, 79, 659-667 (2009).
  78. Rhodium-catalyzed conjugate addition of Sb-aryl-1,5-azastibocines to α,β-unsaturated carbonyl compounds. N. Kakusawa, S. Yasuike and J. Kurita, Heterocycles, 77, 1269-1283 (2009).　
  79. Effect of periodic replacement of the heteroatom on the spectroscopic properties of indole and benzofuran derivatives. A. Muranaka, S. Yasuike, C.-Y. Liu, J. Kurita, N. Kakusawa, T. Tsuchiya, M. Okuda, N. Kobayashi, Y. Matsumoto, K. Yoshida, D. Hashizume and M. Uchiyama, J. Phys. Chem. A., 113, 464-473 (2009).
  80. Palladium-catalyzed carbonylative cross-coupling reaction of triarylantimony dicarboxylates with arylboronic acids: Synthesis of biaryl ketones. W. Qin, S. Yasuike, N. Kakusawa and J. Kurita, J. Organomet. Chem., 693, 2949-2953 (2008).
  81. Triarylantimony dicarboxylates as pseudo-halides for palladium-catalyzed cross-coupling reaction with arylboronic acids triarylbismuthanes without any base. W. Qin, S. Yasuike, N. Kakusawa, Y. Sugawara, M. Kawahata, K. Yamaguchi and J. Kurita, J. Organomet. Chem., 693, 109-116 (2008).
  82. Suzuki-type cross-coupling reaction of pentavalent triarylantimony diacetates with arylboronic acids without a base. S. Yasuike, W. Qin, Y. Sugawara and J. Kurita, Tetrahedron Lett., 48, 719-722 (2007).
  83. A novel transmetallation of triarylstibanes into arylboronate: Boro-induced ipso-deantimonation and its theoretical calculation. S. Yasuike, K. Nakata, W. Qin, T. Kaji and J. Kurita, Chem. Lett., 35, 1402-1403 (2006).
  84. Hypervalent organoantimony compounds 12-ethynyl-tetrahydrodibenz[c,f][1,5]azastibocines: Highly efficient new transmetallating agent for organic halides. N. Kakusawa, Y. Tobiyasu, S. Yasuike, K. Yamaguchi, H. Seki and J. Kurita, J. Organomet. Chem., 691, 2953-2968 (2006).
  85. Synthesis of enantiomerically pure Sb-chirogenic organoantimony compounds and their crystal structures. S. Yasuike, Y. Kishi, S. Kawara, K. Yamaguchi and J. Kurita, J. Organomet. Chem., 691, 2213-2220 (2006).
  86. Synthesis of JOSIPHOS-type ligands via a diastereoselective three-component reaction and their application in asymmetric rhodium-catalyzed hydroborations. S. Yasuike, C. C. Kofink, R. J. Kloetzing, N. Gommermann, K. Tappe, A. Gavryushin and P. Knochel, Tetrahedron: Asymmetry, 16, 3385-3393 (2005).
  87. An organobismuth compound that exhibit cytotoxicity selectively to vascular endothelial cells in vitro. Y. Fujiwara, M. Mitani, S. Yasuike, J. Kurita and T. Kaji, J. Health. Sci., 51, 333-340 (2005).
  88. Catalytic action of triarylstibanes: oxidation of benzoins into benzyls using triarylstibanes under an aerobic condition. S. Yasuike, Y. Kishi, S. Kawara and J. Kurita, Chem. Pharm. Bull., 53, 425-427 (2005).
  89. Cyclic voltammetric study of intramolecular and intermolecular hypervalent organoantimony complexes with Sb…N bonding. K. Hoshino, T. Ogawa, S. Yasuike, H. Seki, J. Kurita, T. Tokunaga and K. Yamaguchi, J. Phys. Chem. B, 108, 18698-18704 (2004).
  90. Non-C2-symmetrical antimony-phosphorus ligand, (R/S)-2-diphenylphosphano-2’-di(p-tolyl)stibano-1,1’-binaphthyl (BINAPSb): preparation and its use for asymmetric reactions as a chiral auxiliary. S. Yasuike, S. Kawara, S. Okajima, H. Seki, K. Yamaguchi and J. Kurita, Tetrahedron Lett., 45, 9135-9138 (2004).
  91. Remarkable reactivity enhancement with Sb---N intra-coordination of ethynyl-1,5-azastibocines in Pd-catalyzed cross-coupling reactions with organic halides. N. Kakusawa, Y. Tobiyasu, S. Yasuike, K. Yamaguchi, H. Seki and J. Kurita, Tetrahedron Lett., 44, 8589-8592 (2003).
  92. A versatile Route to 3-benzoheteroepines containing group 15 and 16 heavier elements involving several novel ring systems, and their thermal stabilities. S. Yasuike, T. Kiharada, T. Tsuchiya and J. Kurita, Chem. Pharm. Bull., 51, 1283-1288 (2003).
  93. 2,2’-Bis(diarylstibano)-1,1’-binaphthyls (BINASbs); a useful chiral ligand for palladium-catalyzed asymmetric allylic alkylation, and the structure of a BINASb-PdCl2 complex. S. Yasuike, S. Okajima, K. Yamaguchi and J. Kurita, Tetrahedron Lett., 44, 6217-6220 (2003).
  94. 光学活性有機アンチモン化合物の合成とその性質に関する研究. 安池修之, Yakugaku Zasshi, 123, 577-585 (2003).
  95. New optically active organoantimony (BINASb) and bismuth (BINABi) compounds comprising a 1,1'-binaphthyl core: synthesis and their use in transition metal-catalyzed asymmetric hydrosilylation of ketones. S. Yasuike, S. Okajima, K. Yamaguchi, H. Seki and J. Kurita, Tetrahedron, 59, 4961-4968 (2003).
  96. Synthesis of Sb-chiral organoantimony compounds having intramolecular Sb…N interaction and their separation into optically pure compounds via ortho-palladated benzylamine complexes. S. Okajima, S. Yasuike, N. Kakusawa, A. Osada, K. Yamaguchi, H. Seki and J. Kurita, J. Organomet. Chem., 656, 234-242 (2002).
  97. Synthesis of optically active organoantimony compounds having an (S)-α-methylbenzyldimethylamine group and its evaluation for asymmetric reaction. S. Yasuike, S. Okajima and J. Kurita, Chem. Pharm. Bull., 50, 1404-1406 (2002).
  98. Synthesis, molecular structure and fluxional behavoir of (R)-7-p-tolyldinaphtho[2,1-b;1’,2’-d]stibole: the first isolated example of optically active group 15 dinaphthoheteroles. S. Yasuike, T. Iida, K. Yamaguchi, H. Seki and J. Kurita, Tetrahedron Lett., 42, 441-444 (2001).
  99. Synthesis of 1-stibaphenalenes, the first example of group 15 phenalenes, via a 1,5-dilithium intermediate. S. Yasuike, M. Niwa, K. Yamaguchi, T. Tsuchiya and J. Kurita, Chem. Lett., 554-555 (2001).
  100. Synthesis and fluxional behavior of dinaphtho[2,1-b;1’,2’-d]-siloles and -germoles, involving the first example of optically active group 14 dinaphthoheterols. S. Yasuike, T. Iida, S. Okajima, K. Yamaguchi, H. Seki and J. Kurita, Tetrahedron, 57, 10047-10053 (2001).
  101. Resolution of racemic Sb-chiral stibindoles using an optically active ortho-palladated benzylamine derivative, via their diastereomeric complexes. J. Kurita, F. Usuda, S. Yasuike, T. Tsuchiya, Y. Tsuda, F. Kiuchi and S, Hosoi, Chem. Commun., 191-192 (2000).
  102. Direct detection of intramolecular Sb…N nonbonded interaction by 1H-13C and 1H-15N heteronuclear multiple bond correlation spectroscopy. T. Tokunaga, H. Seki, S. Yasuike, M. Ikoma, J. Kurita and K. Yamaguchi, Tetrahedron Lett., 41, 1031-1034 (2000).
  103. Synthesis and structure of novel dibenzo[b, i]-1-oxa-6-heteroecines containing group 15 heavier elements. S. Yasuike, S. Tsukada, J. Kurita, T. Tsuchiya, Y. Tsuda, F. Kiuchi and S. Hosoi, Heterocycles, 53, 525-528 (2000).
  104. Confirmation and characterization of the hypervalent Sb…N bonding recognized in triarylstibanes bearing an amino side chain by X-ray, NMR and theoretical caluculations. T. Tokunaga, H. Seki, S. Yasuike, M. Ikoma, J. Kurita and K. Yamaguchi, Tetrahedron, 56, 8833-8839 (2000).
  105. Synthesis and resolution of 2,2’-bis[di(p-tolyl)stibano]-1,1’-binaphthyl (BINASb); the first example of an optically active organoantimony ligand for asymmetric synthesis. S. Yasuike, S. Okajima, K. Yamaguchi, H. Seki and J. Kurita, Tetrahedron: Asymmetry, 11, 4043-4047 (2000).
  106. A versatile synthesis of 1-benzoheteroepines containing group 14, 15, and 16 heavier elements via a common 1,6-dilithium intermediate. S. Yasuike, S. Shiratori, J. Kurita and T. Tsuchiya, Chem. Pharm. Bull., 47, 1108-1114 (1999).
  107. A simple one-pot synthesis of [1]benzotelluro[3,2-b][1]benzotellurophenes and selenium and sulfur analogues from 2,2’-dibromodiphenylacetylene. H. Sashida and S. Yasuike, J. Heterocyclic Chem., 35, 725-726 (1998).
  108. Syntheses of novel group 15 and 16 thieno[2,3-b]-, thieno[3,4-b]-, and thieno[3,2-b]-heteroles. S. Yasuike, J. Kurita and T. Tsuchiya, Heterocycles, 45, 1891-1894 (1997).
  109. Syntheses of novel dithieno[2,3-b;3',2'-f]- and dithieno[3,4-b;3',4'-f]heteroepines containing group 14, 15, and 16 heavier elements. S. Yasuike, F. Nakashima, J. Kurita and T. Tsuchiya, Heterocycles, 45, 1899-1902 (1997).
  110. A versatile synthesis of the group 15 and 16 3-benzoheteropines involving the first isolated examples of several C-unsubstituted 3-benzoheteropines. S. Yasuike, T. Kiharada, J. Kurita and T. Tsuchiya, Chem. Commun., 2183-2184 (1996).
  111. Synthesis of 1-benzometalloles containing group 14, 15 and 16 heavier elements via a common dilithiostyrene intermadiate. J. Kurita, M. Ishii, S. Yasuike and T. Tsuchiya, Chem. Pharm. Bull., 42, 1437-1441 (1994).
  112. Studies on seven-membered heterocycles. XXXIV. Syntheses and reactions 1-benzosilepines, 1-benzogermepines, 1-benzophosphepines, and 1-benzarsepines. S. Shiratori, S. Yasuike, J. Kurita and T. Tsuchiya, Chem. Pharm. Bull., 42, 2441-2448 (1994).
  113. A versatile synthetic route to 1-benzometalloles involing the first examples of several C-unsubstituted benzometalloles. J. Kurita, M. Ishii, S. Yasuike and T. Tsuchiya, J. Chem. Soc., Chem. Commun., 1309-1310 (1993).
  114. Synthesis of the first examples of 1-benzosilepine, 1-benzogermepine, and 1-benzarsepine. J. Kurita, S. Shiratori, S. Yasuike and T. Tsuchiya, Heterocycles, 36, 2677-2680 (1993).
  115. Syntheses of the group 15 1-benzoheteroepines, dibenzo[b,d]heteroepines, and dibenzo[b,f]heteroepines involving the first isolate examples of arsepines and bismepines. S. Yasuike, H. Ohta, S. Shiratori, J. Kurita and T. Tsuchiya, J. Chem. Soc., Chem. Commun., 1817-1819 (1993).
  116. A new route to 1,3-benzoxazepines and 1,3-benzodiazepines via intramolecular Aza-Wittig reaction. J. Kurita, T. Iwata, S. Yasuike and T. Tsuchiya, J. Chem. Soc., Chem. Commun., 81-82 (1992).
  117. Synthesis of first exaples of 1-benzophosphepines. J. Kurita, S. Shiratori, S. Yasuike and T. Tsuchiya, J. Chem. Soc., Chem. Commun., 1227-1228 (1991).
  118. Reaction of pyridazine N-oxides: formation of the first examples of pyrido-oxepines. J. Kurita, N. Kakusawa, S. Yasuike and T. Tsuchiya, Heterocycles, 31, 1937-1940 (1990).

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愛知学院大学
薬学部　薬化学講座
教授：安池修之
講師：松村実生
講師：村田裕基

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愛知県名古屋市千種区楠元町
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愛知学院大学
愛知学院大学薬学部

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