Monday, September 28 | ||
17:00 - | Registration at Grand Court Nagoya | |
18:00 - 20:00 | Opening Session and Welcome Reception - 5th floor of Hotel Grand Court Nagoya (near Kanayama Station) |
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Thuesday, September 29 | ||
8:00 - | Registration |
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8:30 - 8:40 | Opening Remarks Yoshiaki Kawashima (Aichi Gakuin University, Japan) James W. McGinity (University of Texas, USA) |
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Chairs | Pornsak Sriamornsak, Hirofumi Takeuchi | |
8:40 - 9:10 | Plenary Lecture SQUALENOYLATION: A PLATEFORM FOR THE DISCOVERY OF NEW ANTICANCER AND ANTIVIRAL NANOMEDICINES Patric Couvreur, L. Harivardhan Reddy, C. Bourgaux, R. Gref, D. Desmaël, S. Lepêtre, P. Clayette (University Paris-Sud XI and CNRS, France, SPI-BIO, France) |
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Session 1 - Design of novel functional microparticles | ||
9:10 - 9:35 | Invited Lecture -1 DESIGN OF PH-SENSITIVE LIPOSOMES USING POLYMERS Kenji Kono (Osaka Prefecture University, Japan) |
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9:35 - 9:55 | FORMULATION AND CHARACTERISATION OF ORGANIC-INORGANIC
FUNCTIONAL MICROCAPSULES
Yue Long, Jon A. Preece, David York, Zhibing Zhang (University of Birmingham, UK, P&G Technical Centre Ltd., UK) |
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9:55 - 10:15 | STUDY ON THE BREAKING BEHAVIOR OF A MICROCAPSULE Naoki Tsuda, Toshiro Ohtsubo (Sumitomo Chemical Co., Ltd., Japan) |
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10:15 - 10:40 | Break |
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Chairs | Paul W. S. Heng, Hiroshi Yuasa | |
Session 2 - Novel technologies for preparing functional microparticles | ||
10:40 - 11:05 | Invited Lecture -2 CHIMERA AGGLOMERATES FOR EXTRAVASCULAR DELIVERY OF PARTICULATE DRUGS Paolo Colombo (University of Parma, Italy) |
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11:05 - 11:25 | DRUG-LOADED ASCORBYL DIPALMITATE/DSPE-PEG NANOPARTICULATE
SYSTEM Kunikazu Moribe, Sunao Maruyama, Kenjirou Higashi, Keiji Yamamoto (Chiba University, Japan) |
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11:25 - 11:45 | SYNTHESIS OF HIGHLY FUNCTIONALIZED NANOPARTICLES BASED ON
POLY(ALKYL CYANOACRYLATE) BY MEANS OF CLICK CHEMISTRY Benjamin Le Droumaguet, Fethi Bensaid, Juliette Roisin, Karine Andrieux, Patrick Couvreur, Julien Nicolas (Univ. Paris-Sud, France) |
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11:45 - 12:10 | Invited Lecture -3 MICROENCAPSULATED AND RELATED CATALYSTS FOR ORGANIC SYNTHESIS Shū Kobayashi (The University of Tokyo, Japan) |
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Chair | Katsuhide Terada | |
12:25 - 12:55 | Lunch on Seminar -1 (supported by Qualicaps Co. Ltd.) MICROENCAPSULATION BY SPRAY-FREEZE DRYING Hans Leuenberger, Maxim Puchkov, Matthias Plitzko (Ifiip llc, Switzerland, CINCAP GmbH c/o Ifiip llc, Switzerland, Glatt GmbH,Germany) |
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13:05 - 14:25 | Poster & Exhibition -1 |
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Chairs | Alf Lamprecht, Tetsuya Ozeki | |
Session 3 - Microparticles for cancer therapy-1 (supported by Astellas Pharma Inc.) | ||
14:40 - 15:05 | Invited Lecture -4 POLYMERIC MICELLES FOR NANO-COMBINATION DRUG DELIVERY Glen S. Kwon, Ho-Chul Shin, Adam W. G. Alani (University of Wisconsin, USA) |
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15:05 - 15:25 | SODIUM DEOXYCHOLATE INCORPORATING LIPOSOMES FOR HEXAMETHYLMELAMINE (HMM) ORAL DELIVERY: DEVELOPMENT, CHARACTERIZATION AND IN VIVO EVALUATION Yingjie Deng, Jukui Sun, Jinna Cao, Xiaofei Gao, Xiaodong Dong (Shenyang Pharmaceutical University, China) |
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15:25 - 15:45 | LONG-TERM SUSTAINED ANTICANCER EFFECTS OF BIODEGRADABLE MICROSPHERES ENCAPSULATING A SIRNA AGAINST CFLIP OR RAF-1 IN MICE AND RATS BY INDUCING APOPTOSIS Yuuki Takashima, Kosei Toyoshima, Tatsuya Shimizu, Takanori Kanazawa, Hiroaki Okada (Tokyo University of Pharmacy and Life Sciences, Japan) |
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15:45 - 16:10 | Invited Lecture -5 DESIGN OF MELITTIN LOADED PLGA NANOPARTICLES FOR ORAL ADMINISTRATION AND INVESTIGATION OF ANTICANCER EFFICIENCY Fude Cui, Linlin Yang (Shenyang Pharmaceutical University, China) |
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16:10 - 16:35 | Break |
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Chairs | Jörg Kreuter, Yuuki Takashima | |
Session 4 - Microparticles for cancer therapy-2 (supported by Astellas Pharma Inc.) | ||
16:35 - 17:00 | Invited Lecture -6 DELIVERY SYSTEM STRATEGY FOR THE PEGYLATED PEPTIDE AND PROTEIN THERAPEUTICS Tae Hyung Kim, Kang Choon Lee (SungKyunKwan University, Korea) |
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17:00 - 17:20 | INHALABLE NANOFORMULATION FOR TREATMENT OF LUNG CARCINOMA Keishiro Tomoda, Keiji Hirota, Hiroshi Terada, Takehisa Nakajima, Ganeshchandra S. Sonavane, Masahito Komuro, Kenji Kitazato, Kimiko Makino (Tokyo University of Science, Japan) |
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17:20 - 17:45 | Invited Lecture -7 TARGETING OF HIV SANCTUARY SITES USING LIPID BASED ANTIRETROVIRAL NANOCARRIERS Kamalinder K. Singh (S.N.D.T. Women’s University, India) |
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Wednesday, September 30 | ||
Chairs | Glen S. Kwon, Hirokazu Okamoto | |
8:40 - 9:10 | Plenary Lecture SUPRAMOLECULAR ASSEMBLIES OF SMART BLOCK COPOLYMERS AS NANODEVICES FOR GENE AND DRUG DELIVERY Kazunori Kataoka (The University of Tokyo, Japan): |
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Session 5 - Brain targetting with microparticles | ||
9:10 - 9:35 | Invited Lecture -8 DRUG DELIVERY ACROSS THE BLOOD-BRAIN BARRIER TO THE BRAIN USING NANOPARTICLES – RECENT STATUS Jörg Kreuter, Svetlana Gelperina (Goethe-Universität Frankfurt, German, Nanosystem LTD, Russia) |
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9:35 - 10:55 | MALIGNANT BRAIN TUMOR THERAPY IN RATS USING CELL PENETRATION
PEPTIDE - TUMOR SUPPRESSOR PEPTIDE FUSION PEPTIDE, P53P-ANT,
MICROSPHERES Tetsuya Ozeki, Daiki Kaneko, Yoshihiro Imai, Hiroaki Okada (Tokyo University of Pharmacy and Life Sciences, Japan, Nagoya City University, Japan) |
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9:55 - 10:15 | NANOPARTICLES FOR THERAPY OF ALZHEIMER’S DISEASE: ABILITY OF
PEGYLATED POLY(ALKYL CYANOACRYLATE) NANOPARTICLES TO LINK TO THE
Aβ PEPTIDE 1-42 AND TO INFLUENCE ITS AGGREGATION KINETIC Davide Brambilla, Romain Verpillot, Julien Nicolas, Myriam Taverna, Patrick Couvreur, Karine Andrieux (Univ. Paris-Sud, France) |
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10:15 - 10:40 | Break |
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Chairs | Paolo Colombo, Kunikazu Moribe | |
Session 6 - Basic technoilogies for formulating microparticles | ||
10:40 - 11:05 | Invited Lecture -9 PREPARATION OF UNIFORM-SIZED MICROSPHERES AND MICROCAPSULES FOR DRUG DELIVERY Guanghui Ma, Zhiguo Su, Lianyan Wang, Wei Wei, Rong Liu, Qiang Wei (Chinese Academy of Sciences, China) |
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11:05 - 11:25 | MICROENCAPSULATION OF TMBA (1,3,5-TRIMETHYLBARBITURIC ACID) AS BARBITURIC ACID DERIVATIVE BY THE DRYING-IN-LIQUID METHOD IN THE REVERSE EMULSION Kiyomi Fuchigami, Yoshinari Taguchi, Masato Tanaka (Shofu Inc., Japan, Niigata University, Japan) |
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11:25 - 11:50 | Invited Lecture -10 FORMULATION AND PROCESS OPTIMIZATION IN SMALL PARTICLE ENCAPSULATION Paul W. S. Heng, Wun Chyi Chin, Likun Wang, Celine V Liew, Lai Wah Chan (National University of Singapore, Singapore) |
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11:50 - 12:15 | Invited Lecture -11 MICROENCAPSULATION OF SOLID AND LIQUID MODEL CORES AND MORPHOLOGICAL CHARACTERISTICS OF FORMED CAPSULES Hiroyuki Kage, Yoshihide Mawatari, Masato Yamamura (Kyushu Institute of Technology, Japan) |
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Chair | Hiroaki Okada | |
12:25 - 12:55 | Lunch on Seminar -2 (supported by Takeda Pharmaceutical Co. Ltd.) PREPARATION AND PROPERTIES OF MODIFIED RELEASE PELLETS PREPARED BY HOT-MELT EXTRUSION James W. McGinity, Sandra Schilling (University of Texas, USA) | |
13:05 - 14:25 | Poster & Exhibition -2 |
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Mini Symposium -A, B | ||
Room A | Microparticles for oral drug delivery-1 | |
Chairs | Shirui Mao, Hideki Ichikawa | |
14:40 - 15:00 | DEVELOPMENT OF ENTERIC-COATED (S/O) MICROCAPSULES
UTILIZING EDIBLE FATS Kento Kanaya, Masao Sato (Kaneka Co., Japan) |
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15:00 - 15:20 | IMPROVEMENT OF ANTIFUNGAL AND ANTIBACTERIAL ACTIVITY OF INCLUSION
COMPLEXES BETWEEN EUGENOL AND CYCLODEXTRIN Somsak Saesoo, Onanong Nuchuchua, Issara Sramala, Satit Puttipipatkhachorn, Apinan Soottitantawat, Uracha Ruktanonchai (Nantional Science and Technology Developmet Agency, Thailand, Mahidol University, Thailand, Chulalongkorn University, Thailand) |
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15:20 - 15:40 | STUDIES ON MICROENCAPSULATED AND NON-ENCAPSULATED LIPID FORMULATIONS OF BCG
VACCINE IN GUINEA PIGS Allan K. Nadian, Simon Clark, Martin Cross, Julia Vipond, Ann Williams, Mark Chambers, R. Glyn Hewinson, Frank Aldwell (Veterinary Laboratories Agency, UK, Health Protection Agency, UK, University of Otago, New Zealand) |
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15:40 - 16:00 | PREPARATION OF IMMOBILIZED ALLIINASE IN ALGINATE MICROCAPSULES Yeo Lim Lee, Hyun Jin Park (Korea University, Korea) |
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16:00 - 16:25 | Break |
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Room A | Microparticles for oral drug delivery-2 | |
Chairs | Kang Choon Lee, Yuichi Tozuka | |
16:25 - 16:45 | ORAL DELIVERY OF CALCITONIN USING NOVEL NANOPARTICULATE SYSTEM Abdallah M. Makhlof, Martin Werle, Yuichi Tozuka, Hirofumi Takeuchi (Gifu Pharmaceutical University, Japan) |
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16:45 - 17:05 | THE PHYSICAL PROPERTIES OF β-CYCLODEXTRIN INCLUSION COMPLEX CONTAINING LEMONGRASS OIL Wanwisa Srinuanchai, Apinan Soottitantawat, Uracha Ruktanonchai (National Science and Technology Development Agency, Thailand, Chulalongkorn University, Thailand) |
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17:05 - 17:25 | THE PREPARATION OF A NOVEL MULTIPLE CHITOSAN RIBOFLAVIN FLOATING MICROSPHERES USING MICROBUBBLE DISPERSION Lijun Bi, Huimin Yao, Lu Xu, Qifang Wang, Weisan Pan, Zhonggui He, Sanming Li (Shenyang Pharmaceutical University, China) |
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Room B | Microparticles for transmuosal drug delivery-1 | |
Chairs | Yilmaz Capan, Masayuki Yokoyama | |
14:40 - 15:00 | THE DELIVERY OF HYDROPHOBIC COMPOUNDS TO THE RETINA USING
SUBMICRON-SIZED LIPOSOMES Kohei Hironaka, Yuta Inokuchi, Takuya Fujisawa, Yuichi Tozuka, Masamitsu Shimazawa, Hideaki Hara, Hirofumi Takeuchi (Gifu Pharmaceutical University, Japan) |
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15:00 - 15:20 | PHYSICOCHEMICAL STUDY OF NANOCOMPLEXES BETWEEN DICLOFENAC
SODIUM AND THREE TYPES OF CHITOSAN DERIVATIVES AS A NEW CARRIER
FOR OCULAR DELIVERY
Maleenart Petchsangsai, Warayuth Sajomsang, Jutamas Pontrakoon, Uracha Raktanonchai (National Science and Technology Development Agency, Thailand, Mahidol University, Thailand) |
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15:20 - 15:40 | COENZYME Q10-LOADED LIPOSOMES COATED WITH TRIMETHYL CHITOSAN FOR OCULAR ADMINISTRATION PROTECT AGAINST LENS OXIDATIVE DAMAGE IN VITRO AND IN VIVO Jing Zhang, Zhanyou Wang, Tongying Jiang, Siling Wang (Shenyang Pharmaceutical University, China, China Medical University, China) |
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15:40 - 16:00 | THE DEVELOPMENT OF CIPROFLOXACIN DRY POWDERS
FOR PULMONARY DELIVERY M. Miozzi, P. Colombo, Francesca Buttini(University of Parma, Italy) |
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16:00 - 16:25 | Break |
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Room B | Microparticles for transmuosal drug delivery-2 | |
Chairs | Fu-Qiang Hu, Kimiko Makino | |
16:25 - 16:45 | DUAL IMAGING POWDER FOR EVALUATION OF PULMONARY POWDER DELIVERY AND GENE EXPRESSION Hirokazu Okamoto, Tomoyuki Mizuno, Kohta Mohri, Tomoyuki Okuda (Meijo University, Japan) |
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16:45 - 17:05 | EFFECT OF PARTICLE SIZE ON THE IN VITRO-IN VIVO RELEASE OF RESVERATROL FROM PLGA MICROSPHERES Yanjun Wang, Shirui Mao, Wei Sun (Shenyang Pharmaceutical University, China) |
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17:05 - 17:25 | PARENTERAL APPLICATIONS OF NANOCRYSTAL® TECHNOLOGY FOR POORLY WATER SOLUBLE COMPOUNDS Gary G. Liversidge (Elan Drug Technologies) |
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18:30 - | Gala Dinner | |
Thursday, October 1 | ||
Chairs | Valérie Andre-Frei, Yoshie Maitani | |
8:40 - 9:10 | Plenary Lecture NANOTECHNOLOGY AND MICROENCAPSULATION FOR DELIVERY OF “UNDELIVERABLE” DRUGS Vladimir P. Torchilin (Northeastern University, USA) |
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Session 7 - Microparticles for cosmetics-1 (supported by BASF Japan Ltd.) | ||
9:10 - 9:35 | Invited Lecture -12 DEVELOPMENT OF NANOCAPSULE (NC) FOR TRANSDERMAL DELIVERY SYSTEM - CREATION OF NEW PHARMACOLOGIC EFFECTS BY NC BEYOND EXPECTATION - Yoko Yamaguchi , Teruaki Nagasawa, Kayo Matsumoto, Natsumi Nakamura, Kaori Akiyama, Yoshiki Kubota (St. Marianna University, Japan, NANOEGG® Research Laboratories. Inc., Japan) |
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9:35 - 9:55 | THERAPEUTIC PAINT FOR SIMULTANEOUS DELIVERY OF SUCRALFATE GEL AND
CIDOFOVIR IN THE TREATMENT OF VETERINARY VIRAL SKIN INFECTIONS
Gaia Colombo, Alessandra Scagliarini, Laura Gallina, Fabrizio Bortolotti, Enea Menegatti, Paolo Colombo, Fabio Sonvico (University of Ferrara, Italy, University of Bologna, Italy, University of Parma, Italy) |
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9:55 - 10:15 | DEVELOPMENT OF A REDUCED COENZYME Q10-CONTAINING MICROCAPSULE
WITH HIGH STABILITY AGAINST THE OXIDATION IN AIR Shinsuke Akao, Takashi Ueda, Takahiro Ueda (Kaneka Co., Japan) |
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10:15 - 10:40 | Break |
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Chairs | Gaia Colombo, Akihiko Sato | |
Session 8 - Microparticles for cosmetics-2 (supported by BASF Japan Ltd.) | ||
10:40 - 11:00 | SYNTHETIC POLYMER MICELLES IN COSMETICS Kunio Shimada (NOF Corporation, Japan) |
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11:00 - 11:20 | MICROENCAPSULATION: A MARKETING TOOL Pascale Valot (EURACLI, France) |
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11:20 - 11:40 | DEVELOPMENT OF FUNCTIONAL SKIN CARE COSMETICS
USING BIODEGRADABLE PLGA NANOSPHERES H. Tsujimoto, Y. Tsukada, K. Hara,Yohei Bando, N. Miwa, Y. Kawashima (Hosokawa Powder Technology Research Institute, Japan, Prefectural University of Hiroshima, Japan, Aichi Gakuin University, Japan) |
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11:40 - 12:05 | Invited Lecture -13 THERAPEUTIC APPROACHES APPLIED TO COSMETICS: THE CYTOVECTORTM EXAMPLE Bonnet Isabelle, Valérie Andre-Frei, Durieux Florent (BASF Beauty Care Solutions, France) | |
12:05 - 12:15 | Closing Remarks Yilmaz Capan (Hacettepe University, Turkey) |
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12:30 - | Excursion (Tokugawa Art Museum) |